Carisoprodol Overview

Generic Name: Carisoprodol
Drug Class: Skeletal muscle relaxants
Dosage Forms: Tablets (250 mg, 350 mg, 500 mg, 750 mg)

Uses

Carisoprodol is a muscle relaxant that works by blocking pain signals between the nerves and the brain. It is commonly used in combination with rest, physical therapy, and other treatments to relieve pain and discomfort associated with acute musculoskeletal conditions such as muscle spasms, strains, and injuries. Due to its potential for dependency, Carisoprodol is typically prescribed for short-term use, generally 2 to 3 weeks.

Mechanism of Action

Carisoprodol is metabolized in the body to meprobamate, a substance with anxiolytic and sedative properties. The exact mechanism of action is not fully understood, but it is believed to work by interrupting neuronal communication within the reticular formation and spinal cord, resulting in muscle relaxation and relief from pain.

Side Effects

Common Side Effects:

• Drowsiness
• Dizziness
• Headache

Serious Side Effects:

• Allergic Reactions: Hives, difficulty breathing, swelling of the face, lips, tongue, or throat
• Neurological: Seizures (convulsions), confusion, hallucinations
• Serotonin Syndrome: Agitation, hallucinations, fever, sweating, shivering, fast heart rate, muscle stiffness, twitching, loss of coordination, nausea, vomiting, diarrhea
• Overdose Symptoms: Vision problems, confusion, muscle stiffness, loss of coordination, weak or shallow breathing, fainting, seizure, or coma

Note: This is not a complete list of side effects. Always consult your healthcare provider for medical advice about side effects.

Warnings

• Addiction & Dependency: Carisoprodol is habit-forming and can lead to addiction, overdose, or death if misused. It should be used only as prescribed and never shared with others.
• CNS Depression: The medication can impair thinking or reactions, making activities like driving or operating heavy machinery dangerous.
• Withdrawal: Sudden discontinuation after long-term use can lead to withdrawal symptoms. Gradual tapering is recommended under medical supervision.
• Porphyria: Do not use if you have porphyria, a genetic enzyme disorder affecting the nervous system or skin.

Precautions Before Taking

Before using Carisoprodol, inform your doctor if you have:

• Liver disease
• Kidney disease
• A history of seizures

Pregnancy and breastfeeding considerations:

• Pregnancy: The effects on an unborn baby are unknown. Consult your doctor if you are pregnant or planning to become pregnant.
• Breastfeeding: Carisoprodol can pass into breast milk and may cause drowsiness in a nursing baby. Discuss the risks with your doctor.

Age Considerations:

• Not recommended for children under 16 years old.
• Older adults may be more sensitive to the sedative effects of the medication.

Dosage

Usual Adult Dose for Muscle Spasm:

• 250 to 350 mg orally 3 times a day and at bedtime
• Duration: Typically up to 2 to 3 weeks, as long-term use is not recommended due to the potential for dependency.

Missed Dose & Overdose

• Missed Dose: Take the missed dose as soon as you remember, but skip it if it’s almost time for your next dose. Do not double the dose.
• Overdose: Symptoms of overdose include vision problems, confusion, hallucinations, muscle stiffness, loss of coordination, weak or shallow breathing, fainting, seizure, or coma. Seek emergency medical help immediately if an overdose is suspected.

Drug Interactions

Carisoprodol can interact with many medications, including:

• Opioids, sleeping pills, other muscle relaxers, anxiety or seizure medications: Can increase the risk of severe sedation, respiratory depression, or death.
• Other drugs affecting the central nervous system: May exacerbate drowsiness and dizziness.

Always inform your doctor of all medications, including over-the-counter drugs and supplements, to avoid potential interactions.

Storage

Store Carisoprodol at room temperature, away from moisture and heat. Keep it out of reach of children and monitor for any unauthorized use, as it is a controlled substance.

Note: 

The brand name displayed above is specific to this product. Brand names can vary depending on the manufacturer.